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￥ 0.00 renin-angiotensin-aldosterone system (RAAS)
| Catalog No. | Inhibitor Name | AT1 receptor | AT2 receptor | ACE | Renin | RAAS |
|---|---|---|---|---|---|---|
| A11123 | Aliskiren Hemifumarate | *** | ||||
| A10175 | Candesartan | **** | ||||
| A10351 | Enalaprilat Dihydrate | *** | *** | **** | ||
| A10477 | Irbesartan | *** | ||||
| A13201 | PD123319 | * | ||||
| A10710 | Perindopril Erbumine | *** | ||||
| A10176 | Candesartan Cilexetil | **** | ||||
| A10778 | Ramipril | ** | ||||
| A11738 | Captopril | * | ||||
| A16420 | Azilsartan Medoxomil | ** | ||||
| A13747 | Eprosartan Mesylate | **** | ||||
| A11775 | Azilsartan | ** | ||||
| A10905 | Telmisartan | |||||
| A10123 | Benazepril HCl | |||||
| A10350 | Enalapril Maleate | |||||
| A11615 | Olmesartan Medoxomil | |||||
| A11747 | Cilazapril Monohydrate | |||||
| A11876 | Lisinopril | |||||
| A11745 | Moexipril HCl | |||||
| A11749 | Temocapril | |||||
| A11736 | Quinapril HCl | |||||
| A14206 | LCZ696 | |||||
| A11748 | Fosinopril Sodium |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
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Enalapril maleate
Catalog No. A10350 -
Enalaprilat dihydrate
Catalog No. A10351 -
PD 123319 ditrifluoroacetate
Catalog No. A13201 angiotensin AT2 receptor 拮抗剂PD 123319 ditrifluoroacetate是一种有效的，选择性的非肽血管紧张素AT2受体拮抗剂。大鼠肾上腺组织和大脑的IC50值分别为34和210 nM。 了解更多 -
LCZ696 (Valsartan)
Catalog No. A14206 angiotensin receptor-neprilysin 抑制剂LCZ696 (Valsartan)是一种生物利用型双效血管紧张素受体-中性溶血素抑制剂（ARNi），用于治疗高血压和心力衰竭。 了解更多 -
Captopril disulfide
Catalog No. A13521 LTA4 hydrolase 抑制剂Captopril disulfide是LTA4水解酶的可逆竞争性抑制剂（IC50 = 11 M）。Captopril已被证明是血管紧张素转化酶-1（ACE1）的一种，而不是ACE2（IC50 = 22 nM）。 了解更多 -
Angiotensin I (human, mouse, rat)
Catalog No. A14859 Angiotensin I (human,mouse,rat)是由肾素对血管紧张素原的作用形成的。 了解更多 -
Angiotensin III (human, mouse)
Catalog No. A14864 Angiotensin III (human,mouse)是在血管紧张素II的N末端裂解形成的六肽，血管紧张素II是位于红细胞和大多数组织血管床中的血管紧张素酶在肾素-血管紧张素-醛固酮（RAAS）系统中的关键因素。 了解更多 -
Angiotensin 1/2 (1-9)
Catalog No. A14873 Angiotensin 1/2 (1-9)是一种肽（ASP-ARG-VAL-TYR-ILE-HIS-PRO-PHE-HIS），包含从血管紧张素I/II肽转换而来的氨基酸1-9。 了解更多 -
Acetyl Angiotensinogen (1-14), porcine
Catalog No. A14883 Acetyl Angiotensinogen (1-14), porcine血管紧张素原基因编码的蛋白质被称为血管紧张素原或血管紧张素原的前体。 了解更多 -
Angiotensin 1/2 + A (2 - 8)
Catalog No. A14888 Angiotensin 1/2 + A (2 - 8)有效的内源性血管收缩肽；血管紧张素（Ang）的衍生物II。 了解更多 -
VTP-27999 2,2,2-trifluoroacetate
Catalog No. A15281 -
Spinorphin
Catalog No. A15314 -
EXP-3174
Catalog No. A15451 -
MLN-4760
Catalog No. A16884 -
Aliskiren hemifumarate
Catalog No. A11123 -
Candesartan (Atacand)
Catalog No. A10175 RAAS 拮抗剂Candesartan (Atacand)是一种血管紧张素受体阻滞剂（也称为血管紧张素II受体拮抗剂或AIIRA）。 了解更多 -
Benazepril HCl
Catalog No. A10123 -
Clinofibrate
Catalog No. A11184 HMG-CoA Reductase 抑制剂Clinofibrate是一种脂质清除剂，似乎可以改变脂质代谢，减少类固醇诱导的骨细胞内脂质堆积。它还可以有效降低血浆纤维蛋白原水平。抑制hydroxymethylglutaryl coenzyme A reductase (HMGCR)（羟甲基戊二酰辅酶A还原酶），IC50为0.47 mM。 了解更多 -
Rosuvastatin
Catalog No. A11122 -
Irbesartan (Avapro)
Catalog No. A10477 -
Aliskiren (CGP 60536)
Catalog No. A11616 -
Candesartan cilexetil (Atacand)
Catalog No. A10176 Candesartan Cilexetil一种特异性的，非肽类血管生成素II受体（ATR）拮抗剂，也是Candesartan的前体药物，是ATR拮抗剂 了解更多 -
Cilazapril monohydrate
Catalog No. A11747 -
Moexipril hydrochloride
Catalog No. A11745 Moexipril hydrochloride是一种有效的口服活性非巯基血管紧张素转换酶抑制剂(ACE),可作用于高血压和充血性心力衰竭。 了解更多 -
Azilsartan Medoxomil
Catalog No. A16420 angiotensin II receptor type 1 拮抗剂Azilsartan medoxomil是一种口服给药的1型血管紧张素II受体拮抗剂，IC50为0.62 nM。 了解更多 -
Fimasartan
Catalog No. A17477 non-peptide angiotensin II receptor antagonistFimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of angiotensin II, such as systemic vasoconstriction and water retention by the kidneys. 了解更多 -
H-Val-Pro-Pro-OH
Catalog No. A18868 ACE inhibitorH-Val-Pro-Pro-OH, a milk-derived proline peptides derivative, is an inhibitor of Angiotensin I converting enzyme (ACE), with an IC50 of 9 μM. 了解更多 -
Zofenopril
Catalog No. A13615 ACE inhibitorZofenopril is an angiotensin-converting enzyme (ACE) inhibitor with an IC50 of 81 μM. 了解更多 -
Imidaprilate
Catalog No. A20003 ACE inhibitorImidaprilate is an active metabolite of TA-6366, acts as a potent angiotensin converting enzyme (ACE) inhibitor, with an IC50 of 2.6 nM, and is used in the research of hypertensive disease. 了解更多 -
Azilsartan medoxomil monopotassium
Catalog No. A20860 angiotensin II receptor type 1 antagonistAzilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. 了解更多 -
Sparsentan
Catalog No. A20879 angiotensin II and endothelin A receptor antagonistSparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. 了解更多 -
Lisinopril
Catalog No. A21064 angiotensin-converting enzyme inhibitorLisinopril (MK-521) is angiotensin-converting enzyme inhibitor, used in treatment of hypertension, congestive heart failure, and heart attacks. 了解更多 -
Losartan (D4 Carboxylic Acid)
Catalog No. A21578 angiotensin II receptor antagonistLosartan D4 Carboxylic Acid is the deuterium labeled Losartan(EXP-3174), which is an angiotensin II receptor antagonist. 了解更多 -
Azilsartan D5
Catalog No. A21600 angiotensin II type 1 receptor antagonistAzilsartan D5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. 了解更多 -
Fosinopril sodium
Catalog No. A11748 -
Lisinopril (Zestril)
Catalog No. A11876 Lisinopril (Zestril)是血管紧张素转换酶抑制剂，用于治疗高血压，充血性心力衰竭和心脏病发作，还用于预防糖尿病的肾和视网膜并发症。 了解更多
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