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￥ 0.00 FAK
| Catalog No. | Inhibitor Name | FAK | Other |
|---|---|---|---|
| A12580 | PF-00562271 | **** | CDK2/CyclinE,CDK3/CyclinE,CDK1/CyclinB |
| A11192 | PF-562271 | **** | CDK2/CyclinE,CDK3/CyclinE,CDK1/CyclinB |
| A11235 | PF-573228 | * | |
| A11507 | TAE226 | ** | Insulin Receptor,IGF-1R,c-Met |
| A11171 | PF-03814735 | * | Aurora A,Aurora B,FLT1 |
| A11142 | PF-431396 | ** | |
| A13140 | PND-1186 | **** | |
| A11929 | Defactinib | ||
| A15543 | CEP-37440 | ** | ALK |
| A15765 | GSK2256098 | **** |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
10 个项目
每页
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PF-03814735
Catalog No. A11171 Aurora A/B Kinase 抑制剂PF-03814735是一种新颖，有效且可逆的Aurora A/B抑制剂，IC50为0.8 nM/5 nM，对Flt3，FAK，TrkA的效力较低，对Met和FGFR1的活性最低。 了解更多 -
PF-4618433
Catalog No. A13461 -
PF-00562271
Catalog No. A12580 FAK 抑制剂PF-00562271是PF-562271的苯磺酸盐，是一种有效的，ATP竞争性，可逆的FAK和Pyk2抑制剂，IC50分别为1.5 nM和14 nM。 了解更多 -
PF-04554878 (Defactinib)
Catalog No. A11929 FAK 抑制剂PF-04554878 (Defactinib)是一种新型FAK激酶抑制剂，可降低胰腺神经内分泌肿瘤细胞的生长并诱导其凋亡。 了解更多 -
NVP-TAE 226
Catalog No. A11507 FAK 抑制剂NVP-TAE 226是一种强效FAK抑制剂，IC50为5.5 nM，对pyk2(IC50=3.5 nM)有适度的强效作用；对InsR, IGF-1R, ALK和c-Met的效力降低10-100倍。 了解更多
10 个项目
每页
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