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Epigenetic Reader Domain

Epigenetic Reader Domain

Inhibitory Selectivity

Catalog No.	Inhibitor Name	Epigenetic Reader Domain
A12729	(*)-JQ1	***
A11783	I-BET151	*
A12545	PFI-1	**
A11440	I-BET-762	***
A13956	RVX-208	*
A13227	SGC-CBP30	****
A13163	Bromosporine	****
A13890	OTX015	****
A12948	UNC1215	**
A13717	UNC669	*
A14133	GSK1324726A	***
A13749	MS436	**
A13068	CPI-203	***
A13957	PFI-3

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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Selective BRD9 抑制剂

I-BRD9是一种有效的选择性BRD9抑制剂，pIC50为7.3，而对BRD4的pIC50为5.3。了解更多

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BI-7273

Catalog No. A16068
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BRD9 BD 抑制剂

BI-7273是一种选择性的，细胞可渗透的BRD9 BD抑制剂。了解更多

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Catalog No. A13163
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bromodomain 抑制剂

Bromosporine是一种针对溴结构域的广谱抑制剂，对于BRD2，BRD4，BRD9和CECR2的IC50分别为0.41μM，0.29μM，0.122μM和0.017μM。了解更多

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BI-9564

Catalog No. A16196
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