Epigenetic Reader Domain
Catalog No. | Inhibitor Name | Epigenetic Reader Domain |
---|---|---|
A12729 | (*)-JQ1 | *** |
A11783 | I-BET151 | * |
A12545 | PFI-1 | ** |
A11440 | I-BET-762 | *** |
A13956 | RVX-208 | * |
A13227 | SGC-CBP30 | **** |
A13163 | Bromosporine | **** |
A13890 | OTX015 | **** |
A12948 | UNC1215 | ** |
A13717 | UNC669 | * |
A14133 | GSK1324726A | *** |
A13749 | MS436 | ** |
A13068 | CPI-203 | *** |
A13957 | PFI-3 |
Notes:
1.Hover mouse over " " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
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Bromosporine
Catalog No. A13163 bromodomain 抑制剂Bromosporine是一种针对溴结构域的广谱抑制剂,对于BRD2,BRD4,BRD9和CECR2的IC50分别为0.41μM,0.29μM,0.122μM和0.017μM。 了解更多 -
I-BRD9
Catalog No. A15872