IKK/IκB

Inhibitory Selectivity

Catalog No.	Inhibitor Name	IκB	IKK	Other
A11957	BAY 11-7082	*		E2-conjugating enzymes
A12836	IKK-16		***
A11579	TPCA-1		****
A12559	BMS-345541		**
A12746	SC-514		**	CDK2/CyclinA,AUR2,PRAK
A12470	Bay 11-7085	*
A12789	PS-1145		***
A15488	LY2409881		****
A11148	BX-795			PDK-1,c-Kit,CDK2/CyclinE
A12837	IMD 0354
A11323	Bardoxolone Methyl			NF-κB,Nrf2
A15900	AZD3264
A12953	WS6			EBP1
A12952	WS3			EBP1
A11318	BMS-345541 HCl		**
A11339	Bay 65-1942	*
A11485	MRT67307		**	TBK1
A13108	PHA 408
A15171	MLN120B

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.