Protein Kinase C (PKC)
Catalog No. | Inhibitor Name | PKC | PKCα | PKCβ | PKCγ | PKCδ | PKCε | PKCζ | PKCη | PKCθ | PKCμ | Other |
---|---|---|---|---|---|---|---|---|---|---|---|---|
A10356 | Enzastaurin | ** | *** | * | * | |||||||
A11554 | Sotrastaurin | **** | **** | **** | **** | **** | **** | |||||
A10864 | Staurosporine | **** | **** | ** | * | * | **** | c-Fgr,phosphorylase kinase,S6 kinase | ||||
A13790 | Go 6983 | *** | *** | *** | *** | ** | * | |||||
A13197 | Bisindolylmaleimide I | ** | *** | ** | PDGFR | |||||||
A13514 | Ro 31-8220 Mesylate | **** | *** | ** | ** | |||||||
A12650 | Midostaurin | ** | ** | ** | * | * | * | * | PPK,KDR,c-Syk | |||
A12419 | Go6976 | *** | **** | *** | FLT3,JAK2 | |||||||
A10766 | Quercetin | Sirtuin,Src,PI3Kγ | ||||||||||
A10616 | Myricitrin | |||||||||||
A10196 | Chelerythrine chloride | * | ||||||||||
A10261 | Bryostatin 1 | *** | ||||||||||
A10286 | Daphnetin | * | EGFR, PKA | |||||||||
A12399 | Ruboxistaurin (LY333531) | * | **** | * | * | ** | ||||||
A14871 | PKC (19-36) | * |
Notes:
1.Hover mouse over " " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
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Prostratin
Catalog No. A13679 -
(-)-Indolactam V
Catalog No. A13043 PKC activator(-)-Indolactam V是一种蛋白激酶C激活剂,可将人ES细胞衍生的定形内胚层强有力地引导至胰腺内胚层中。 了解更多 -
12-O-tetradecanoyl phorbol-13-acetate
Catalog No. A14616 PKC activator12-O-tetradecanoyl phorbol-13-acetate是佛波醇的二酯,是从巴豆油中提取的促肿瘤化合物。它是在体内和体外以nM浓度可逆的高效蛋白激酶C(PKC)激活剂。 了解更多