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￥ 0.00 FGFR
| Catalog No. | Inhibitor Name | FGFR | FGFR1 | FGFR2 | FGFR3 | FGFR4 | Other |
|---|---|---|---|---|---|---|---|
| A10080 | Ponatinib | **** | Abl,PDGFRα,VEGFR2 | ||||
| A11159 | BGJ398 | **** | **** | **** | ** | VEGFR2,Lyn,Kit | |
| A10137 | Nintedanib | ** | ** | ** | * | VEGFR3,VEGFR2,LCK | |
| A10703 | PD173074 | ** | VEGFR2,c-Src | ||||
| A11411 | Dovitinib | *** | *** | FLT3,c-Kit,VEGFR3/FLT4 | |||
| A11075 | AZD4547 | **** | **** | **** | * | KDR,IGFR | |
| A10715 | Danusertib | ** | Aurora A,Abl,TrkA | ||||
| A10953 | Orantinib | * | PDGFRβ,Flk1 | ||||
| A10254 | Brivanib | * | VEGFR2,Flk1,VEGFR1 | ||||
| A10198 | Dovitinib Dilactic Acid | *** | *** | FLT3,c-Kit,VEGFR3/FLT4 | |||
| A11753 | MK-2461 | ** | ** | ** | |||
| A10162 | Brivanib Alaninate | * | VEGFR2,Flk1,VEGFR1 | ||||
| A13211 | SSR128129E | * | VEGFR2,PDGFRβ | ||||
| A11558 | SU5402 | ** | |||||
| A15534 | BLU9931 | * | * | * | **** | ||
| A12357 | FIIN-2 | **** | *** | ** | ** | FLT3,c-Kit,VEGFR3/FLT4 | |
| A14415 | CH5183284 | *** | *** | *** | * | VEGFR2 | |
| A11244 | LY2874455 | **** | **** | *** | *** | ||
| A15957 | Erdafitinib | ||||||
| A10508 | KW-2449 | ** | FLT3, Bcr-Abl, Aurora A, PDGFRβ, IGF-1R, EGFR | ||||
| A10699 | Pazopanib HCl | * | VEGFR1, VEGFR2, VEGFR3, PDGFR, c-Kit, c-Fms | ||||
| A11518 | Pazopanib | * | VEGFR1, VEGFR2, VEGFR3, PDGFR, c-Kit, c-Fms | ||||
| A13111 | R 1530 | * | Chk2, KDR, FGFR, Aurora A, Cdk2, VEGFR-2, PDGFRβ | ||||
| A15073 | E-3810 | *** | ** | VEGFR1, VEGFR2, VEGFR3 | |||
| A15848 | FIIN-3 | *** | ** | ** | ** | ||
| A15957 | Alofanib (RPT835) |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
12 个项目
每页
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Dovitinib Dilactic acid (TKI258 Dilactic acid)
Catalog No. A10198 RTK 抑制剂Dovitinib是一种小分子多靶点酪氨酸激酶抑制剂，可抑制通过ZNF198-FGFR1或BCR-FGFR1转化为IL3独立性的Ba / F3细胞，IC50值分别为150 nM和90 nM。 了解更多 -
Debio-1347 (CH5183284)
Catalog No. A14415 FGFR1/2/3 抑制剂Debio-1347 (CH5183284)是成纤维细胞生长因子受体亚型1（FGFR-1），2（FGFR-2）和3（FGFR-3）的生物利用抑制剂，具有潜在的抗肿瘤活性。 了解更多 -
LY 2874455
Catalog No. A11244 -
FIIN-2
Catalog No. A12357 -
NVP-BGJ398 phosphate
Catalog No. A15194 FGFR 抑制剂NVP-BGJ398 phosphate是一种新型的选择性泛特异性FGFR抑制剂，对FGFR1，FGFR2和FGFR3的IC50分别为0.9、1.4和1 nM。与FGFR4和VEGFR2相比，对FGFR具有40倍以上的选择性，并且对Abl，Fyn，Kit，Lck，Lyn和Yes的活性很小。 了解更多 -
Dovitinib (TKI-258)
Catalog No. A11411 RTK 抑制剂Dovitinib是一种小分子多靶点酪氨酸激酶抑制剂，可抑制通过ZNF198-FGFR1或BCR-FGFR1转化为IL3独立性的Ba / F3细胞，IC50值分别为150 nM和90 nM。 了解更多 -
FIIN-3
Catalog No. A15848 -
Nintedanib esylate
Catalog No. A16197 RTK 抑制剂Nintedanib esylate是多种受体酪氨酸激酶（RTK）和非受体酪氨酸激酶（nRTK）的有效抑制剂。 了解更多 -
BGJ398 (NVP-BGJ398)
Catalog No. A11159 FGFR 抑制剂BGJ398 (NVP-BGJ398)是一种有效的选择性抑制剂，具有成纤维细胞生长因子受体（FGFR）酪氨酸激酶1、2、3和4的潜在抗血管生成和抗肿瘤活性（对于FGFR1，FGFR2，FGFR3，IC50值为0.9、1.4、1.0和60 nM， 和FGFR4）。 了解更多
12 个项目
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