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TGF-β / Smad Inhibitors

TGF-β / Smad Inhibitors

Inhibitory Selectivity

Catalog No.	Inhibitor Name	ALK1	ALK2	ALK3	ALK4	TGFβRI/ALK5	ALK6	ALK7	TGFβRII	TGF-β	Other
A10826	SB431542					**
A11205	LDN-193189		****	***
A11017	Galunisertib					**
A11133	LY2109761					***			*
A10827	SB525334					***
A11157	SB505124				**	**
A11083	GW788388					***
A13446	LY364947					**			*		RIPK2,CK1δ,MLK-7K
A11762	RepSox					****
A11478	LDN-193189 HCl		****	***
A14311	K02288	****	****	***	*	*	****
A16096	LDN-214117		***
A14066	SD-208					**
A14213	EW-7197				***	****
A14298	ML347	**	***	*			*
A12821	LDN-212854	****	****	**	*	*
A12820	DMH1		**
A16209	Pirfenidone
A10449	Hesperetin										Histamine receptor
A12358	A 83-01				***	**		****
A12924	ITD 1									*
A14436	A 77-01					***
A16065	SIS3
A16207	R-268712					****

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.