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￥ 0.00 PDGFR
| Catalog No. | Inhibitor Name | PDGFR | PDGFRα | PDGFRβ | Other |
|---|---|---|---|---|---|
| A10001 | Sorafenib Tosylate | ** | ** | Raf-1,VEGFR2/Flk1,B-Raf | |
| A10468 | Imatinib Mesylate | c-Kit,v-Abl | |||
| A10880 | Sunitinib Malate | **** | FLT3,Kit,VEGFR2 | ||
| A10080 | Ponatinib | **** | Abl,VEGFR2,FGFR1 | ||
| A10103 | Axitinib | *** | **** | VEGFR1/FLT1,VEGFR2/Flk1,VEGFR3 | |
| A10259 | Imatinib | ** | c-Kit,v-Abl | ||
| A10137 | Nintedanib | ** | ** | VEGFR3,VEGFR2,LCK | |
| A10699 | Pazopanib HCl | ** | VEGFR1,VEGFR2,VEGFR3 | ||
| A11411 | Dovitinib | * | *** | FLT3,c-Kit,FGFR1 | |
| A10025 | Linifanib | ** | VEGFR1/FLT1,CSF-1R,FLT3 | ||
| A11052 | Crenolanib | **** | **** | ||
| A10558 | Masitinib | * | * | Kit,Lyn B,Abl1 | |
| A10101 | Tivozanib | *** | ** | VEGFR2,VEGFR3,EphB2 | |
| A10610 | Amuvatinib | *** | c-Kit (D816H),FLT3 (D835Y) | ||
| A10608 | Motesanib Diphosphate | ** | VEGFR1,VEGFR2,VEGFR3 | ||
| A10953 | Orantinib | *** | FGFR1,Flk1 | ||
| A11350 | CP-673451 | *** | **** | c-Kit,VEGFR2,VEGFR1 | |
| A10502 | Ki8751 | ** | VEGFR2,c-Kit,FGFR2 | ||
| A10903 | Telatinib | *** | c-Kit,VEGFR3,VEGFR2 | ||
| A11207 | PP121 | **** | Hck,VEGFR,mTOR | ||
| A11518 | Pazopanib | ** | VEGFR1,VEGFR2,VEGFR3 | ||
| A10504 | KRN 633 | * | * | VEGFR3,VEGFR2,VEGFR1 | |
| A10198 | Dovitinib Dilactic Acid | * | *** | FLT3,c-Kit,VEGFR3/FLT4 | |
| A11753 | MK-2461 | *** | c-Met (M1250T),c-Met (Y1235D),c-Met (Y1230H) | ||
| A14156 | AZD2932 | **** | Flt3,VEGFR-2,c-Kit | ||
| A15062 | DCC-2618 | *** | *** | c-Kit |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
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Pazopanib (GW-786034)
Catalog No. A11518 VEGFR 抑制剂Pazopanib (GW-786034)是VEGFR-1，VEGFR-2，VEGFR-3，PDGFR-a/β和c-kit的有效且选择性的多靶点酪氨酸激酶抑制剂，可阻止肿瘤生长并抑制血管生成。 了解更多
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