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HDAC

Inhibitory Selectivity

Catalog No.Inhibitor Name HDAC HDAC1 HDAC2 HDAC3 HDAC4HDAC5 HDAC6 HDAC7 HDAC8 HDAC9 HDAC10 HDAC11 HD1 HD2
A10979Vorinostat
****
A10611Entinostat
**
*
A10518Panobinostat
****
A10947Trichostatin A
****
A10586Mocetinostat
**
**
*
*
A10122Belinostat
***
A11920Romidepsin
***
***
A10560MC1568
*
A11042Tubastatin A HCl
*
***
A10488Givinostat
****
****
A10516Dacinostat
***
A10246CUDC-101
****
****
***
****
***
***
****
**
**
**
***
A10830Pracinostat
***
**
***
***
***
*
**
**
**
***
**
A11152PCI-34051
*
*
****
*
A10337Droxinostat
*
*
*
A10700Abexinostat
****
***
****
***
**
***
A13218RGFP966
**
A11037AR-42
***
A11940Ricolinostat
**
***
***
*
*
****
*
**
A11964Tacedinaline
*
*
*
**
A11153CUDC-907
****
****
****
**
*
***
**
**
****
****
A11355M344
**
A10954Tubacin
****
A13139RG2833
***
****
A12556Resminostat
***
***
**
A15489BRD73954
*
***
**
A11361BG45
*
*
**
A143544SC-202
*
*
*
A16431CAY10603
**
****
A14341LMK-235
***
****
A14032Nexturastat A
****
A14128TMP269
**
**
***
***
A14197HPOB
*
*
*
***
*
*
A12722Scriptaid
A12616Tasquinimod
A11042Tubastatin A
***

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

23 个项目

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  1. KD 5170
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    KD 5170

    Catalog No. A15354
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    HDAC 抑制剂
    KD 5170是一种新型的基于巯基酮的组蛋白脱乙酰基酶抑制剂，在体外和体内均表现出广谱的抗肿瘤活性。 了解更多
  2. CAY10603
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    CAY10603

    Catalog No. A16431
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    HDAC6 抑制剂
    CAY10603是一种有效的选择性HDAC6抑制剂，IC50为2 pM，选择性是其他HDAC的200倍以上。 了解更多
  3. Tubastatin A
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    Tubastatin A

    Catalog No. A16770
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    HDAC6 inhibitor
    Tubastatin A is a potent and selective HDAC6 inhibitor with IC50 of 15 nM in a cell-free assay, and is selective (1000-fold more) against all other isozymes except HDAC8 (57-fold more). 了解更多
  4. Trichostatin-A (TSA)
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    Trichostatin-A (TSA)

    Catalog No. A10947
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    HDAC 抑制剂
    Trichostatin-A (TSA)是抑制HDAC 1、3、4、6和10，IC50值约为20 nM。 了解更多
  5. ACY-1215 (Rocilinostat)
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    ACY-1215 (Rocilinostat)

    Catalog No. A11940
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    HDAC6 抑制剂
    ACY-1215 (Rocilinostat)是一种选择性HDAC6抑制剂，从而通过Hsp90的超乙酰化作用破坏Hsp90蛋白伴侣系统，并防止随后的总蛋白降解。 了解更多
  6. BRD73954
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    BRD73954

    Catalog No. A15489
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    HDAC 抑制剂
    BRD73954是一种小分子抑制剂，可有效抑制HDAC6和HDAC8（IC50分别为36和120 nM）。 了解更多
  7. ACY-738
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    ACY-738

    Catalog No. A15934
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    HDAC6 抑制剂
    ACY-738是一种有效的选择性HDAC6抑制剂，具有改善的脑生物利用度。ACY-738抑制HDAC6的纳摩尔浓度低，选择性比I类HDAC高60到1500倍。 了解更多
  8. CUDC-907 (Fimepinostat)
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    CUDC-907 (Fimepinostat)

    Catalog No. A11153
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    PI3K/HDAC 抑制剂
    CUDC-907 (Fimepinostat)是针对PI3K和HDAC的单一小分子抑制剂，作用于PI3Kα和HDAC1/2/3/10，IC50分别为19 nM和1.7 nM/5 nM/1.8 nM/2.8 nM。 了解更多
  9. TCS HDAC6 20b
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    TCS HDAC6 20b

    Catalog No. A15387
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    HDAC6 抑制剂
    TCS HDAC6 20b是组蛋白脱乙酰基酶6（HDAC6）的选择性抑制剂。与紫杉醇联合抑制HCT116的生长。还抑制雌激素刺激的MCF-7细胞的生长。 了解更多
  10. Droxinostat
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    Droxinostat

    Catalog No. A10337
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    HDAC 抑制剂
    Droxinostat是HDAC3，HDAC6和HDAC8的选择性抑制剂，显示出可比较的HDAC6和HDAC8抑制作用，IC50分别为2.47和1.46μmol/ L。 了解更多
  11. BRD9757
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    BRD9757

    Catalog No. A12911
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    HDAC6 抑制剂
    BRD9757是一种高效且选择性的HDAC6抑制剂，对HDAC6的IC50为30 nM。 了解更多
  12. Resminostat hydrochloride
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    Resminostat hydrochloride

    Catalog No. A15220
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    HDAC 抑制剂
    Resminostat hydrochloride是HDAC1/3/6的有效抑制剂（IC50 = 43-72 nM）；对HDAC8的效力较低，IC50为877 nM。 了解更多
  13. BG45
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    BG45

    Catalog No. A11361
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    HDAC 抑制剂
    BG45是一种HDAC I类抑制剂，对HDAC3具有选择性（IC50 = 289 nM）。它抑制HDAC1，HDAC2和HDAC6的效力大大降低（IC50分别为2、2和> 20μM）。 了解更多
  14. Tubacin
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    Tubacin

    Catalog No. A10954
    HDAC6 抑制剂
    Tubacin (tubulin acetylation inducer)是一种高效且选择性强，可逆，可透过细胞的HDAC6抑制剂，IC50为4 nM。 了解更多
  15. Citarinostat (ACY-241)
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    Citarinostat (ACY-241)

    Catalog No. A12758
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    HDAC6 抑制剂
    ACY-241是HDAC6的新型，选择性和口服抑制剂。对HDAC6和HDAC3的IC50分别为2.6 nM和46 nM。 了解更多
  16. Tubastatin A HCl
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    Tubastatin A HCl

    Catalog No. A11042
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    HDAC6 抑制剂
    Tubastatin A HCl是一种有效的选择性HDAC6抑制剂，在无细胞试验中IC50为15 nM。它对除HDAC8（57倍）以外的所有其他同工酶（1000倍）具有选择性。 了解更多
  17. Resminostat
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    Resminostat

    Catalog No. A12556
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    HDAC 抑制剂
    Resminostat，也称为RAS2410，是一种有效的I和II类组蛋白脱乙酰基酶（HDAC）抑制剂。它结合并抑制HDAC，从而导致高度乙酰化的组蛋白的积累。选择性的抑制HDAC1/3/6，IC50为42.5 nM/50.1 nM/71.8 nM，作用于HDAC8效果弱，IC50为877 nM。 了解更多
  18. SW-100
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    SW-100

    Catalog No. A18947
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    HDAC6 inhibitor
    SW-100, a selective histone deacetylase 6 (HDAC6) inhibitor with an IC50 of 2.3 nM, shows at least 1000-fold selectivity for HDAC6 relative to all other HDAC isozymes. 了解更多
  19. Nexturastat A
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    Nexturastat A

    Catalog No. A14032
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    HDAC6 抑制剂
    Nexturastat A是一种芳基脲衍生物，可作为组蛋白脱乙酰基酶6（HDAC6）的有效且高度选择性的抑制剂（IC50 = 5.02+/-0.60 nM）。 了解更多
  20. SKLB-23bb
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    SKLB-23bb

    Catalog No. A18339
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    HDAC6 inhibitor
    SKLB-23bb is a potent and selective inhibitor for HDAC6 with an IC50 of 17 nM and shows 25-fold and 200-fold selectivity relative to HDAC1 (IC50=422 nM) and HDAC8 (IC50=3398 nM), respectively. 了解更多
  21. ACY-775
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    ACY-775

    Catalog No. A12456
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    HDAC6 inhibitor
    ACY-775 is a potent and selective inhibitor of the of histone deacetylase 6 (HDAC6) with an IC50 of 7.5?nM. 了解更多
  22. HPOB
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    HPOB

    Catalog No. A14197
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    HDAC6 抑制剂
    HPOB是组蛋白去乙酰化酶6(HDAC6；IC50 = 56 nM)。 了解更多
  23. SS-208
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    SS-208

    Catalog No. A18952
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    HDAC6 inhibitor
    SS-208 is a selective HDAC6 inhibitor, with an IC50 of 12 nM. SS-208 possesses anti-tumor activity in melanoma. 了解更多

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